epigenetic modulators of bromodomain proteins

Bromodomain proteins play an integral role in the regulation of transcription and chromatin remodeling by acting as readers of acetylated histone lysine residues. Active Motif offers small molecules to study the effect of changes in bromodomain activity.

Name Appl. Format Cat No. Price  
JQ1 (+/-) BET Bromodomain Inhibitor 25 mg 14066 $400 Buy
5 mg 14067 $125 Buy
RVX-208 BET Bromodomain Antagonist 25 mg 14090 $305 Buy
5 mg 14091 $90 Buy